Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ α-Amyloid Precursor Protein Modulator
A cell-permeable benzolactam derived PKC activator (K
MilliporeSigma™ Calbiochem™ UbcH13 Inhibitor, NSC697923
The UbcH13 Inhibitor, NSC697923 controls the biological activity of UbcH13. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ 2-Chloro-2'-deoxyadenosine
A deoxyadenosine analog that displays strong antileukemic and immunosuppressive activity.
MilliporeSigma™ Calbiochem™ 5-Nitro-2-(3-phenylpropylamino)benzoic Acid
Potent Cl- channel blocker (IC50 = 100 nM-100 μM), depending on channel subtype and assay method.
MilliporeSigma™ Calbiochem™ Gemcitabine, HCl
A bioavailable, moderately toxic, deoxyctytidine analog with anti-metabolite and anti-tumor properties
MilliporeSigma™ Calbiochem™ Adenovirus Proteinase Inhibitor, NSC 37249
An inhibitor of adenovirus cysteine proteinase AVP that simultaneously targets AVP co-factor pVIc N-terminal binding pocket (K
MilliporeSigma™ Calbiochem™ TLR8 Agonist, cpd14b
A potent agonist of Toll-like receptor 8 agonist (TLR8, EC50 = 200 nM).
MilliporeSigma™ Calbiochem™ Granzyme B Inhibitor I
The Granzyme B Inhibitor I controls the biological activity of Granzyme B. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ Wnt Antagonist III, Box5
The Wnt Antagonist III, Box5 controls the biological activity of Wnt. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ Kir6.2/SUR1 Channel Activator, VU0071063
A fast acting, reversible, and selective activator of Kir6.2/SUR1 channels (EC50 = 7 μM).
MilliporeSigma™ Calbiochem™ LYP Inhibitor II, LTV-1
The LYP Inhibitor II, LTV-1 controls the biological activity of LYP. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Myristoylated-FEEERA, mP6
A cell-permeable myristoylated hexapeptide that selectively inhibits integrin outside-in signaling without affecting inside-out signaling. Blocks the interaction of Gα3 and integrin β3 subunit.
MilliporeSigma™ Calbiochem™ NMDAR2C/2D Inhibitor, DQP-1105
The NMDAR2C/2D Inhibitor, DQP-1105 controls the biological activity of NMDAR2C/2D. This small molecule/inhibitor is primarily used for Neuroscience applications.
MilliporeSigma™ Calbiochem™ Caspase-1/4 Inhibitor, VX-765
A cell-permeable prodrug that upon conversion to its active form inhibits caspase-1 and 4 activity (Ki = 800 pM and 600 pM, respectively).